Dermorphin 5mg
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Dermorphin
Dermorphin is an opioid peptide originally found in the skin of amphibians; it exhibits analgesic and antinociceptive activities, acting as an agonist at μ-opioid receptors (μORs). In animal models of thermal, mechanical, and chemical pain, dermorphin increases pain thresholds.
Product Info
Cas No. 77614-16-5
Purity ≥96%
Formula C40H50N8O10
Formula Wt. 802.88
Chemical Name
Tyrosyl-alanyl-phenylalanyl-glycyl-tyrosyl-prolyl-serinamide
IUPAC Name
(2S)-N-[(2S)-1-amino-3-hydroxy-1-oxopropan-2-yl]-1-[(2S)-2-[[2-[[(2S)-2- [[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl] amino]-3-phenylpropanoyl]amino]acetyl]amino]-3-(4-hydroxyphenyl) propanoyl]pyrrolidine-2-carboxamide
Solubility Slightly soluble in water.
Appearance
White to off white powder
Shipping And Storage
Store Temp
-20°C
Ship Temp
Ambient
Refrences
Mizoguchi H, Bagetta G, Sakurada T, et al. Dermorphin tetrapeptide analogs as potent and long-lasting analgesics with pharmacological profiles distinct from morphine. Peptides. 2011 Feb;32(2):421-7. PMID: 21126548. Guzevatykh LS, Voronina TA, Emel’ianova TG, et al. Comparative analysis of analgesic activities of dermorphin, [DPro6]-dermorphin, and their C-terminal tripeptides. Izv Akad Nauk Ser Biol. 2007 Sep-Oct;(5):577-82. PMID: 18038625.STORAGE INSTRUCTION:
All of Our Products are manufactured using the Lyophilization (Freeze Drying) process, which ensures that our products remain 100% stable for shipping for up to 24-36 month.
Once the peptides are reconstituted (mixed with bacteriostatic water), they just be stored in the fridge to maintain stability After reconstitution, the peptides will remain stable for up to 30 days.
Lyophilization is a unique dehydration process, also known as cryodesiccation, where the peptides are frozen and then subjected to low pressure. This causes the water in the peptide vial to sublimate directly from solid to gas, leaving behind a stable, crystalline white structure known as lyophilized peptide The puffy white powder can be stored at room temperature until you’re ready to reconstitute it with bacteriostatic water.
Once peptides have been received, it is imperative that they are kept cold and away from light. If the peptides will be used immediately, or in the next several days, weeks or months short-term refrigeration under 4c (39F) is generally acceptable. Lyophilized peptides are usually stable at room temperatures for several weeks or more, so if they will be utilized within weeks or months such storage is typically adequate.
However, for longer term storage (several months to years) it is more preferable to store peptides in a freezer at -80C (-112F).
When storin peptides for months or even years, freezing is optimal in order to preserve the peptide’s stability.
COMING SOON!!!
Dermorphin
Dermorphin is an opioid peptide originally found in the skin of amphibians; it exhibits analgesic and antinociceptive activities, acting as an agonist at μ-opioid receptors (μORs). In animal models of thermal, mechanical, and chemical pain, dermorphin increases pain thresholds.
Product Info
Cas No. 77614-16-5
Purity ≥96%
Formula C40H50N8O10
Formula Wt. 802.88
Chemical Name
Tyrosyl-alanyl-phenylalanyl-glycyl-tyrosyl-prolyl-serinamide
IUPAC Name
(2S)-N-[(2S)-1-amino-3-hydroxy-1-oxopropan-2-yl]-1-[(2S)-2-[[2-[[(2S)-2- [[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl] amino]-3-phenylpropanoyl]amino]acetyl]amino]-3-(4-hydroxyphenyl) propanoyl]pyrrolidine-2-carboxamide
Solubility Slightly soluble in water.
Appearance
White to off white powder
Shipping And Storage
Store Temp
-20°C
Ship Temp
Ambient
Refrences
Mizoguchi H, Bagetta G, Sakurada T, et al. Dermorphin tetrapeptide analogs as potent and long-lasting analgesics with pharmacological profiles distinct from morphine. Peptides. 2011 Feb;32(2):421-7. PMID: 21126548. Guzevatykh LS, Voronina TA, Emel'ianova TG, et al. Comparative analysis of analgesic activities of dermorphin, [DPro6]-dermorphin, and their C-terminal tripeptides. Izv Akad Nauk Ser Biol. 2007 Sep-Oct;(5):577-82. PMID: 18038625.STORAGE INSTRUCTION:
All of Our Products are manufactured using the Lyophilization (Freeze Drying) process, which ensures that our products remain 100% stable for shipping for up to 24-36 month.
Once the peptides are reconstituted (mixed with bacteriostatic water), they just be stored in the fridge to maintain stability After reconstitution, the peptides will remain stable for up to 30 days.
Lyophilization is a unique dehydration process, also known as cryodesiccation, where the peptides are frozen and then subjected to low pressure. This causes the water in the peptide vial to sublimate directly from solid to gas, leaving behind a stable, crystalline white structure known as lyophilized peptide The puffy white powder can be stored at room temperature until you're ready to reconstitute it with bacteriostatic water.
Once peptides have been received, it is imperative that they are kept cold and away from light. If the peptides will be used immediately, or in the next several days, weeks or months short-term refrigeration under 4c (39F) is generally acceptable. Lyophilized peptides are usually stable at room temperatures for several weeks or more, so if they will be utilized within weeks or months such storage is typically adequate.
However, for longer term storage (several months to years) it is more preferable to store peptides in a freezer at -80C (-112F).
When storin peptides for months or even years, freezing is optimal in order to preserve the peptide's stability.
COMING SOON!!!
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